Oligomerization and allosteric modulation in G -protein coupled receptors / edited by Terry Kenakin

Includes bibliographical references and index

Approaches for probing allosteric interactions at 7 transmembrane spanning receptors / Michael T. Klein, Paige N. Vinson, Colleen M. Niswender -- Pharmacology of metabotropic glutamate receptor allosteric modulators: structural basis and therapeutic potential for CNS disorders / Karen J. Gregory, Meredith J. Noetzel, Colleen M. Niswender -- Mining the potential of label-free biosensors for seven-transmembrane receptor drug discovery / Magalie Rocheville, Julio Martin, Jeff Jerman, Evi Kostenis -- G protein-coupled receptors in cancer: biochemical interactions and drug design / Yves Audigier, François-Xavier Picault, Carline Chaves-Almagro, Bernard Masri -- GPCRs in stem cell function / Van A. Doze, Dianne M. Perez -- Application of receptor theory to allosteric modulation of receptors / David A. Hall -- What ligand-gated ion channels can tell us about the allosteric regulation of G protein-coupled receptors / Frederick J. Ehlert -- Modeling cooperativity effects in dimeric G protein-coupled receptors / Jesús Giraldo -- Chemokine receptor oligomerization and allostery / Bryan Stephens, Tracy M. Handel -- Fine-tuning of GPCR signals by intracellular G protein modulators / Peishen Zhao, Wendy Cladman, Hubert H.M. Van Tol, Peter Chidiac