Oligomerization and allosteric modulation in G -protein coupled receptors / edited by Terry Kenakin - First edition - xiii, 471 pages, 8 unnumbered pages of plates : illustrations (some color) ; 24 cm - Progress in molecular biology and translational science, v. 115 1877-1173 ; . - Progress in molecular biology and translational science ; v. 115 .

Includes bibliographical references and index

Approaches for probing allosteric interactions at 7 transmembrane spanning receptors / Pharmacology of metabotropic glutamate receptor allosteric modulators: structural basis and therapeutic potential for CNS disorders / Mining the potential of label-free biosensors for seven-transmembrane receptor drug discovery / G protein-coupled receptors in cancer: biochemical interactions and drug design / GPCRs in stem cell function / Application of receptor theory to allosteric modulation of receptors / What ligand-gated ion channels can tell us about the allosteric regulation of G protein-coupled receptors / Modeling cooperativity effects in dimeric G protein-coupled receptors / Chemokine receptor oligomerization and allostery / Fine-tuning of GPCR signals by intracellular G protein modulators / Michael T. Klein, Paige N. Vinson, Colleen M. Niswender -- Karen J. Gregory, Meredith J. Noetzel, Colleen M. Niswender -- Magalie Rocheville, Julio Martin, Jeff Jerman, Evi Kostenis -- Yves Audigier, François-Xavier Picault, Carline Chaves-Almagro, Bernard Masri -- Van A. Doze, Dianne M. Perez -- David A. Hall -- Frederick J. Ehlert -- Jesús Giraldo -- Bryan Stephens, Tracy M. Handel -- Peishen Zhao, Wendy Cladman, Hubert H.M. Van Tol, Peter Chidiac

0123945879 9780123945877


G proteins--Receptors
Allosteric regulation

572 / PRO